β-Tosylethylamine: A Useful Reagent for Preparation of N-Protected Amides, Carbamates, and Related Compounds. Application to Synthesis of β-Lactams

Darren DiPietro, Robert M. Borzilleri, Steven M. Weinreb

Research output: Contribution to journalArticle

29 Citations (Scopus)

Abstract

Readily prepared β-tosylethylamine (3) can be used to synthesize N-tosylethyl (TSE)-protected amido compounds and β-lactams, which can be deprotected under mild conditions with potassium tert-butoxide.

Original languageEnglish (US)
Pages (from-to)5856-5857
Number of pages2
JournalJournal of Organic Chemistry
Volume59
Issue number20
DOIs
StatePublished - Oct 1 1994

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Lactams
Carbamates
Amides
potassium tert-butoxide

All Science Journal Classification (ASJC) codes

  • Organic Chemistry

Cite this

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β-Tosylethylamine : A Useful Reagent for Preparation of N-Protected Amides, Carbamates, and Related Compounds. Application to Synthesis of β-Lactams. / DiPietro, Darren; Borzilleri, Robert M.; Weinreb, Steven M.

In: Journal of Organic Chemistry, Vol. 59, No. 20, 01.10.1994, p. 5856-5857.

Research output: Contribution to journalArticle

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