A point mutation that confers constitutive activity to CXCR4 reveals that T140 is an inverse agonist and that AMD3100 and ALX40-4C are weak partial agonists

Wen Bo Zhang, Jean Marc Navenot, Bodduluri Haribabu, Hirokazu Tamamuraz, Kenichi Hiramatu, Akane Omagari, Gang Pei, John P. Manfredi, Nobutaka Fujii, James R. Broach, Stephen C. Peiper

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