A simple, rapid and efficient protocol for the selective phosphorylation of phenols with dibenzyl phosphite

Lee Jonathan Silverberg, John L. Dillon, Purushotham Vemishetti

Research output: Contribution to journalArticle

67 Citations (Scopus)

Abstract

Phosphorylation of phenols with dibenzyl phosphite, carbon tetrachloride, N,N-diisopropylethylamine, and catalytic DMAP in acetonitrile at -10°C is rapid, mild, clean, high yielding, and selective.

Original languageEnglish (US)
Pages (from-to)771-774
Number of pages4
JournalTetrahedron Letters
Volume37
Issue number6
DOIs
StatePublished - Feb 5 1996

Fingerprint

Phosphites
Phosphorylation
Carbon Tetrachloride
Phenols
acetonitrile
N,N-diisopropylethylamine

All Science Journal Classification (ASJC) codes

  • Biochemistry
  • Drug Discovery
  • Organic Chemistry

Cite this

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title = "A simple, rapid and efficient protocol for the selective phosphorylation of phenols with dibenzyl phosphite",
abstract = "Phosphorylation of phenols with dibenzyl phosphite, carbon tetrachloride, N,N-diisopropylethylamine, and catalytic DMAP in acetonitrile at -10°C is rapid, mild, clean, high yielding, and selective.",
author = "Silverberg, {Lee Jonathan} and Dillon, {John L.} and Purushotham Vemishetti",
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A simple, rapid and efficient protocol for the selective phosphorylation of phenols with dibenzyl phosphite. / Silverberg, Lee Jonathan; Dillon, John L.; Vemishetti, Purushotham.

In: Tetrahedron Letters, Vol. 37, No. 6, 05.02.1996, p. 771-774.

Research output: Contribution to journalArticle

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AU - Dillon, John L.

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AB - Phosphorylation of phenols with dibenzyl phosphite, carbon tetrachloride, N,N-diisopropylethylamine, and catalytic DMAP in acetonitrile at -10°C is rapid, mild, clean, high yielding, and selective.

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